Llwytho...

Functionalized Scout Fragments for Site-Specific Covalent Ligand Discovery and Optimization

[Image: see text] Covalent ligands are a versatile class of chemical probes and drugs that can target noncanonical sites on proteins and display differentiated pharmacodynamic properties. Chemical proteomic methods have been introduced that leverage electrophilic fragments to globally profile the co...

Disgrifiad llawn

Wedi'i Gadw mewn:
Manylion Llyfryddiaeth
Cyhoeddwyd yn:ACS Cent Sci
Prif Awduron: Crowley, Vincent M., Thielert, Marvin, Cravatt, Benjamin F.
Fformat: Artigo
Iaith:Inglês
Cyhoeddwyd: American Chemical Society 2021
Mynediad Ar-lein:https://ncbi.nlm.nih.gov/pmc/articles/PMC8155467/
https://ncbi.nlm.nih.gov/pubmed/34056091
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acscentsci.0c01336
Tagiau: Ychwanegu Tag
Dim Tagiau, Byddwch y cyntaf i dagio'r cofnod hwn!