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Characterization of Direct Perturbations on Voltage-Gated Sodium Current by Esaxerenone, a Nonsteroidal Mineralocorticoid Receptor Blocker

Esaxerenone (ESAX; CS-3150, Minnebro(®)) is known to be a newly non-steroidal mineralocorticoid receptor (MR) antagonist. However, its modulatory actions on different types of ionic currents in electrically excitable cells remain largely unanswered. The present investigations were undertaken to expl...

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Publicado en:Biomedicines
Main Authors: Chang, Wei-Ting, Wu, Sheng-Nan
Formato: Artigo
Idioma:Inglês
Publicado: MDPI 2021
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC8153305/
https://ncbi.nlm.nih.gov/pubmed/34068333
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/biomedicines9050549
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