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ABT-199 inhibits Hedgehog pathway by acting as a competitive inhibitor of oxysterol, rather as a BH3 mimetic

Aberrantly activated Hedgehog (Hh) pathway is critical for driving the initiation and progression of multiple types of cancers, including medulloblastoma (MB) and basal cellular carcinoma (BCC). The majority of current Hh antagonist function by targeting the transmembrane domain of the oncoprotein S...

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Dettagli Bibliografici
Pubblicato in:Acta Pharmacol Sin
Autori principali: Wang, Juan, Zhang, Yu, Huang, Wen-jing, Yang, Jun, Tang, Wei-guo, Huang, Tao-min, Tan, Wen-fu
Natura: Artigo
Lingua:Inglês
Pubblicazione: Springer Singapore 2020
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC8149392/
https://ncbi.nlm.nih.gov/pubmed/32855528
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/s41401-020-00504-4
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