Lataa...

Physiologically‐based pharmacokinetic modeling to predict drug interactions of lemborexant with CYP3A inhibitors

Lemborexant, a recently approved dual orexin receptor antagonist for treatment of adults with insomnia, is eliminated primarily by cytochrome P450 (CYP)3A metabolism. The recommended dose of lemborexant is 5 mg once per night, with a maximum recommended dose of 10 mg once daily. A physiologically‐ba...

Täydet tiedot

Tallennettuna:
Bibliografiset tiedot
Julkaisussa:CPT Pharmacometrics Syst Pharmacol
Päätekijät: Ueno, Takashi, Miyajima, Yukiko, Landry, Ishani, Lalovic, Bojan, Schuck, Edgar
Aineistotyyppi: Artigo
Kieli:Inglês
Julkaistu: John Wiley and Sons Inc. 2021
Aiheet:
Linkit:https://ncbi.nlm.nih.gov/pmc/articles/PMC8129715/
https://ncbi.nlm.nih.gov/pubmed/33704920
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/psp4.12606
Tagit: Lisää tagi
Ei tageja, Lisää ensimmäinen tagi!