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Human fetal liver metabolism of oxycodone is mediated by CYP3A7

Oxycodone is an opioid analgesic that is commonly prescribed to pregnant women to treat moderate to severe pain. It has been shown to cross the placenta and distribute to the fetus. Oxycodone is mainly metabolized by CYP3A4 in adult liver. Since CYP3A7 is abundantly expressed in the fetal liver and...

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Publicado en:AAPS J
Main Authors: Shum, Sara, Isoherranen, Nina
Formato: Artigo
Idioma:Inglês
Publicado: 2021
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC8106324/
https://ncbi.nlm.nih.gov/pubmed/33438174
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1208/s12248-020-00537-x
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