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Disulfiram Abrogates Morphine Tolerance—A Possible Role of µ-Opioid Receptor-Related G-Protein Activation in the Striatum

One of the key strategies for effective pain management involves delaying analgesic tolerance. Early clinical reports indicate an extraordinary effectiveness of off-label disulfiram—an agent designed for alcohol use disorder—in potentiating opioid analgesia and abrogation of tolerance. Our study aim...

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Detalhes bibliográficos
Publicado no:Int J Mol Sci
Main Authors: de Corde-Skurska, Anna, Krzascik, Pawel, Lesniak, Anna, Sacharczuk, Mariusz, Nagraba, Lukasz, Bujalska-Zadrozny, Magdalena
Formato: Artigo
Idioma:Inglês
Publicado em: MDPI 2021
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC8071001/
https://ncbi.nlm.nih.gov/pubmed/33919998
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/ijms22084057
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