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Gender-based differences in brain and plasma pharmacokinetics of letrozole in sprague-dawley rats: Application of physiologically-based pharmacokinetic modeling to gain quantitative insights

Based on the discovery that the estrogen synthase aromatase (CYP19A1) is abundantly expressed in high- grade gliomas, the aromatase inhibitor, letrozole is being investigated in pre-clinical models as a novel agent against this malignancy. Here, we investigated the systemic and brain pharmacokinetic...

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Veröffentlicht in:PLoS One
Hauptverfasser: Arora, Priyanka, Gudelsky, Gary, Desai, Pankaj B.
Format: Artigo
Sprache:Inglês
Veröffentlicht: Public Library of Science 2021
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Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC8018653/
https://ncbi.nlm.nih.gov/pubmed/33798227
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1371/journal.pone.0248579
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