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Design of pyrido[2,3-d]pyrimidin-7-one inhibitors of receptor interacting protein kinase-2 (RIPK2) and nucleotide-binding oligomerization domain (NOD) cell signaling

Receptor interacting protein kinase-2 (RIPK2) is an enzyme involved in the transduction of pro-inflammatory nucleotide-binding oligomerization domain (NOD) cell signaling, a pathway implicated in numerous chronic inflammatory conditions. Herein, a pyrido[2,3-d]pyrimidin-7-one based class of RIPK2 ki...

詳細記述

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書誌詳細
出版年:Eur J Med Chem
主要な著者: Nikhar, Sameer, Siokas, Ioannis, Schlicher, Lisa, Lee, Seungheon, Gyrd-Hansen, Mads, Degterev, Alexei, Cuny, Gregory D.
フォーマット: Artigo
言語:Inglês
出版事項: 2021
主題:
オンライン・アクセス:https://ncbi.nlm.nih.gov/pmc/articles/PMC8009825/
https://ncbi.nlm.nih.gov/pubmed/33601309
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.ejmech.2021.113252
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