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Explainable Deep Relational Networks for Predicting Compound–Protein Affinities and Contacts

Predicting compound–protein affinity is beneficial for accelerating drug discovery. Doing so without the often-unavailable structure data is gaining interest. However, recent progress in structure-free affinity prediction, made by machine learning, focuses on accuracy but leaves much to be desired f...

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Podrobná bibliografie
Vydáno v:J Chem Inf Model
Hlavní autoři: Karimi, Mostafa, Wu, Di, Wang, Zhangyang, Shen, Yang
Médium: Artigo
Jazyk:Inglês
Vydáno: 2020
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC7987499/
https://ncbi.nlm.nih.gov/pubmed/33347301
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jcim.0c00866
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