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1,4-Substituted Triazoles as Nonsteroidal Anti-Androgens for Prostate Cancer Treatment

Prostate cancer (PC) is the fifth leading cause of cancer death in men, and the androgen receptor (AR) represents the primary target for PC treatment, even though the disease frequently progresses toward androgen-independent forms. Most of the commercially available nonsteroidal antiandrogens show a...

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Detalles Bibliográficos
Publicado en:J Med Chem
Autores principales: Ferroni, Claudia, Pepe, Antonella, Kim, Yeong Sang, Lee, Sunmin, Guerrini, Andrea, Parenti, Marco Daniele, Tesei, Anna, Zamagni, Alice, Cortesi, Michela, Zaffaroni, Nadia, De Cesare, Michelandrea, Beretta, Giovanni Luca, Trepel, Jane B., Malhotra, Sanjay V., Varchi, Greta
Formato: Artigo
Lenguaje:Inglês
Publicado: 2017
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC7983173/
https://ncbi.nlm.nih.gov/pubmed/28272894
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jmedchem.7b00105
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