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Human ATP-binding cassette transporters ABCB1 and ABCG2 confer resistance to histone deacetylase 6 inhibitor ricolinostat (ACY-1215) in cancer cell lines

Ricolinostat is the first orally available, selective inhibitor of histone deacetylase 6 (HDAC6), currently under evaluation in clinical trials in patients with various malignancies. It is likely that the inevitable emergence of resistance to ricolinostat is likely to reduce its clinical effectivene...

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Dettagli Bibliografici
Pubblicato in:Biochem Pharmacol
Autori principali: Wu, Chung-Pu, Hsieh, Ya-Ju, Murakami, Megumi, Vahedi, Shahrooz, Hsiao, Sung-Han, Yeh, Ni, Chou, An-Wei, Li, Yan-Qing, Wu, Yu-Shan, Yu, Jau-Song, Ambudkar, Suresh V.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2018
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7983170/
https://ncbi.nlm.nih.gov/pubmed/30028995
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bcp.2018.07.018
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