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α,γ-Dioxygenated amides via tandem Brook rearrangement/radical oxygenation reactions and their application to syntheses of γ-lactams

Pyrrolidones are common heterocyclic fragments in various biologically active compounds. Here, a two-step radical-based approach to γ-lactams bearing three to four stereocenters starting from epoxides, N-allylic silylacetamides and TEMPO is reported. The sequence starts with a new tandem nucleophili...

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Dettagli Bibliografici
Pubblicato in:Beilstein J Org Chem
Autori principali: Klychnikov, Mikhail K, Pohl, Radek, Císařová, Ivana, Jahn, Ullrich
Natura: Artigo
Lingua:Inglês
Pubblicazione: Beilstein-Institut 2021
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7961876/
https://ncbi.nlm.nih.gov/pubmed/33777244
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3762/bjoc.17.58
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