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Inhibitory mechanism of reveromycin A at the tRNA binding site of a class I synthetase

The polyketide natural product reveromycin A (RM-A) exhibits antifungal, anticancer, anti-bone metastasis, anti-periodontitis and anti-osteoporosis activities by selectively inhibiting eukaryotic cytoplasmic isoleucyl-tRNA synthetase (IleRS). Herein, a co-crystal structure suggests that the RM-A mol...

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Gorde:
Xehetasun bibliografikoak
Argitaratua izan da:Nat Commun
Egile Nagusiak: Chen, Bingyi, Luo, Siting, Zhang, Songxuan, Ju, Yingchen, Gu, Qiong, Xu, Jun, Yang, Xiang-Lei, Zhou, Huihao
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: Nature Publishing Group UK 2021
Gaiak:
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC7955072/
https://ncbi.nlm.nih.gov/pubmed/33712620
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/s41467-021-21902-0
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