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Furin-Mediated Self-Assembly of Olsalazine Nanoparticles for Targeted Raman Imaging of Tumors

Olsalazine (Olsa) is a broad-spectrum anti-cancer agent acting as a DNA methylation inhibitor. When conjugated to 2-cyano-6-aminobenzothiazole and a peptide substrate specific for the tumor-overexpressed enzyme furin, it can self-assemble into nanoparticles that can be detected by chemical exchange...

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Dades bibliogràfiques
Publicat a:Angew Chem Int Ed Engl
Autors principals: Yuan, Yue, Raj, Piyush, Zhang, Jia, Siddhanta, Soumik, Barman, Ishan, Bulte, Jeff W.M.
Format: Artigo
Idioma:Inglês
Publicat: 2021
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC7902394/
https://ncbi.nlm.nih.gov/pubmed/33325142
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/anie.202014839
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