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Synthesis of trifluoromethyl ketones by nucleophilic trifluoromethylation of esters under a fluoroform/KHMDS/triglyme system

A straightforward method that enables the formation of biologically attractive trifluoromethyl ketones from readily available methyl esters using the potent greenhouse gas fluoroform (HCF(3), HFC-23) was developed. The combination of fluoroform and KHMDS in triglyme at −40 °C was effective for this...

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Bibliographic Details
Published in:Beilstein J Org Chem
Main Authors: Fujihira, Yamato, Liang, Yumeng, Ono, Makoto, Hirano, Kazuki, Kagawa, Takumi, Shibata, Norio
Format: Artigo
Language:Inglês
Published: Beilstein-Institut 2021
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Online Access:https://ncbi.nlm.nih.gov/pmc/articles/PMC7884878/
https://ncbi.nlm.nih.gov/pubmed/33633811
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3762/bjoc.17.39
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