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Discovery of New Catalytic Topoisomerase II Inhibitors for Anticancer Therapeutics

Poison inhibitors of DNA topoisomerase II (TOP2) are clinically used drugs that cause cancer cell death by inducing DNA damage, which mechanism of action is also associated with serious side effects such as secondary malignancy and cardiotoxicity. In contrast, TOP2 catalytic inhibitors induce limite...

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Dettagli Bibliografici
Pubblicato in:Front Oncol
Autori principali: Matias-Barrios, Victor M., Radaeva, Mariia, Song, Yi, Alperstein, Zaccary, Lee, Ahn R., Schmitt, Veronika, Lee, Joseph, Ban, Fuqiang, Xie, Ning, Qi, Jianfei, Lallous, Nada, Gleave, Martin E., Cherkasov, Artem, Dong, Xuesen
Natura: Artigo
Lingua:Inglês
Pubblicazione: Frontiers Media S.A. 2021
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7883873/
https://ncbi.nlm.nih.gov/pubmed/33598437
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3389/fonc.2020.633142
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