A carregar...

Tryptophan-75 Is a Low-Energy Channel-Gating Residue that Facilitates Substrate Egress/Access in Cytochrome P450 2D6

CYP2D6 is a major drug metabolizing enzyme with a buried active site. Channels leading to the active site from various enzyme surfaces are believed to facilitate ligand egress and access to the active site. The present study used molecular dynamics (MD) and in vitro studies with CYP2D6*1 and a Trp75...

ver descrição completa

Na minha lista:
Detalhes bibliográficos
Publicado no:Drug Metab Dispos
Main Authors: McCarty, Kevin D., Ratliff, Samuel A., Furge, Kyle A., Furge, Laura Lowe
Formato: Artigo
Idioma:Inglês
Publicado em: The American Society for Pharmacology and Experimental Therapeutics 2021
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC7883074/
https://ncbi.nlm.nih.gov/pubmed/33376147
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/dmd.120.000274
Tags: Adicionar Tag
Sem tags, seja o primeiro a adicionar uma tag!