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Exploring 1-adamantanamine as an alternative amine moiety for metabolically labile azepane ring in newly synthesized benzo[d]thiazol-2(3H)one σ receptor ligands

In this work we report the structure-activity relationships, binding properties, and metabolic stability studies of a series of benzo[d]thiazol-2(3H)one as sigma receptors (σRs) ligands. Specifically, to improve the metabolic stability of the cyclic amine fragment of our lead compound (SN56), the me...

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Detalhes bibliográficos
Publicado no:Med Chem Res
Main Authors: Intagliata, Sebastiano, Agha, Hebaalla, Kopajtic, Theresa A., Katz, Jonathan L., Kamble, Shyam H., Sharma, Abhisheak, Avery, Bonnie A., McCurdy, Christopher R.
Formato: Artigo
Idioma:Inglês
Publicado em: 2020
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Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC7880169/
https://ncbi.nlm.nih.gov/pubmed/33584084
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s00044-020-02597-2
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