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Druggable Transient Pockets in Protein Kinases

Drug discovery using small molecule inhibitors is reaching a stalemate due to low selectivity, adverse off-target effects and inevitable failures in clinical trials. Conventional chemical screening methods may miss potent small molecules because of their use of simple but outdated kits composed of r...

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Detalhes bibliográficos
Publicado no:Molecules
Main Authors: Umezawa, Koji, Kii, Isao
Formato: Artigo
Idioma:Inglês
Publicado em: MDPI 2021
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC7865889/
https://ncbi.nlm.nih.gov/pubmed/33513739
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/molecules26030651
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