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Inhibitors targeting Bruton’s tyrosine kinase in cancers: drug development advances

Bruton’s tyrosine kinase (BTK) inhibitor is a promising novel agent that has potential efficiency in B-cell malignancies. It took approximately 20 years from target discovery to new drug approval. The first-in-class drug ibrutinib creates possibilities for an era of chemotherapy-free management of B...

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Publicat a:Leukemia
Autors principals: Wen, Tingyu, Wang, Jinsong, Shi, Yuankai, Qian, Haili, Liu, Peng
Format: Artigo
Idioma:Inglês
Publicat: Nature Publishing Group UK 2020
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC7862069/
https://ncbi.nlm.nih.gov/pubmed/33122850
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/s41375-020-01072-6
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