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EGFR/ErbB2-Targeting Lapatinib Therapy for Aggressive Prolactinomas

CONTEXT: Approximately 10% to 20% of prolactinomas are resistant to dopamine agonist therapy. The ErbB signaling pathway may drive aggressive prolactinoma behavior. OBJECTIVE: We evaluated lapatinib, an ErbB1-epidermal growth factor receptor (EGFR)/ErbB2 or human EGFR2 (HER2) tyrosine kinase inhibit...

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Detalhes bibliográficos
Publicado no:J Clin Endocrinol Metab
Main Authors: Cooper, Odelia, Bonert, Vivien S, Rudnick, Jeremy, Pressman, Barry D, Lo, Janet, Salvatori, Roberto, Yuen, Kevin C J, Fleseriu, Maria, Melmed, Shlomo
Formato: Artigo
Idioma:Inglês
Publicado em: Oxford University Press 2020
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC7823257/
https://ncbi.nlm.nih.gov/pubmed/33150390
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1210/clinem/dgaa805
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