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The Bicyclic Form of galacto-Noeurostegine Is a Potent Inhibitor of β-Galactocerebrosidase

[Image: see text] Competitive inhibitors of galactocerebrosidase (GALC) could be candidates for pharmacological chaperone therapy of patients with Krabbe disease. The known and selective nortropane-type iminosugar galacto-noeurostegine has been found to competitively inhibit GALC with K(i) = 7 μM at...

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Bibliografske podrobnosti
izdano v:ACS Med Chem Lett
Main Authors: Viuff, Agnete, Salamone, Stéphane, McLoughlin, Joseph, Deane, Janet E., Jensen, Henrik H.
Format: Artigo
Jezik:Inglês
Izdano: American Chemical Society 2020
Online dostop:https://ncbi.nlm.nih.gov/pmc/articles/PMC7812600/
https://ncbi.nlm.nih.gov/pubmed/33488964
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acsmedchemlett.0c00377
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