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DIPG-71. SELECTIVE HDAC INHIBITOR RG2833 INDUCES DIPG CELL DEATH VIA DOWNREGULATION OF THE NFĸB PATHWAY

Histone deacetylase (HDAC) inhibitor panobinostat demonstrated activity against diffuse intrinsic pontine glioma (DIPG) in vitro, but its efficacy in vivo was limited by toxicity and poor blood brain barrier penetration. RG2833 (RGFP109) is a selective HDAC1/3 inhibitor that has established brain pe...

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Détails bibliographiques
Publié dans:Neuro Oncol
Auteurs principaux: Barnett, Katherine, Novak, Orlandi, Eberhart, Charles, Raabe, Eric
Format: Artigo
Langue:Inglês
Publié: Oxford University Press 2020
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC7715076/
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1093/neuonc/noaa222.113
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