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Novel 1-Amidino-4-Phenylpiperazines as Potent Agonists at Human TAAR1 Receptor: Rational Design, Synthesis, Biological Evaluation and Molecular Docking Studies

Targeting trace amine-associated receptor 1 (TAAR1) receptor continues to offer an intriguing opportunity to develop innovative therapies in different pharmacological settings. Pursuing our endeavors in the search for effective and safe human TAAR1 (hTAAR1) ligands, we synthesized a new series of 1-...

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Detalhes bibliográficos
Publicado no:Pharmaceuticals (Basel)
Main Authors: Francesconi, Valeria, Cichero, Elena, Kanov, Evgeny V., Laurini, Erik, Pricl, Sabrina, Gainetdinov, Raul R., Tonelli, Michele
Formato: Artigo
Idioma:Inglês
Publicado em: MDPI 2020
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC7697893/
https://ncbi.nlm.nih.gov/pubmed/33202687
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/ph13110391
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