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Evaluation of Actinium-225 Labeled Minigastrin Analogue [(225)Ac]Ac-DOTA-PP-F11N for Targeted Alpha Particle Therapy

The overexpression of cholecystokinin B receptor (CCKBR) in human cancers led to the development of radiolabeled minigastrin analogues for targeted radionuclide therapy, which aims to deliver cytotoxic radiation specifically to cancer cells. Alpha emitters (e.g., actinium-225) possess high potency i...

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Dettagli Bibliografici
Pubblicato in:Pharmaceutics
Autori principali: Qin, Yun, Imobersteg, Stefan, Blanc, Alain, Frank, Stephan, Schibli, Roger, Béhé, Martin P., Grzmil, Michal
Natura: Artigo
Lingua:Inglês
Pubblicazione: MDPI 2020
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7696055/
https://ncbi.nlm.nih.gov/pubmed/33198403
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/pharmaceutics12111088
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