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Structural Basis for Activation of Human Sirtuin 6 by Fluvastatin

[Image: see text] Sirtuins are NAD(+)-dependent protein lysine deacylases that are considered attractive drug targets for aging-related diseases. Sirt6 deacetylates, e.g., transcription factors and histone H3, and regulates metabolic processes and stress responses. It has been implicated in lifespan...

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Detalhes bibliográficos
Publicado no:ACS Med Chem Lett
Main Authors: You, Weijie, Steegborn, Clemens
Formato: Artigo
Idioma:Inglês
Publicado em: American Chemical Society 2020
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC7667847/
https://ncbi.nlm.nih.gov/pubmed/33214841
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acsmedchemlett.0c00407
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