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Histone Deacetylase Inhibitors as Multitarget-Directed Epi-Drugs in Blocking PI3K Oncogenic Signaling: A Polypharmacology Approach

Genetic mutations and aberrant epigenetic alterations are the triggers for carcinogenesis. The emergence of the drugs targeting epigenetic aberrations has provided a better outlook for cancer treatment. Histone deacetylases (HDACs) are epigenetic modifiers playing critical roles in numerous key biol...

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Detalhes bibliográficos
Publicado no:Int J Mol Sci
Main Authors: Ranganna, Kasturi, Selvam, Chelliah, Shivachar, Amruthesh, Yousefipour, Zivar
Formato: Artigo
Idioma:Inglês
Publicado em: MDPI 2020
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC7662987/
https://ncbi.nlm.nih.gov/pubmed/33147762
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/ijms21218198
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