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Crystal Structure of the Kinase Domain of MerTK in Complex with AZD7762 Provides Clues for Structure-Based Drug Development

Aberrant tyrosine-protein kinase Mer (MerTK) expression triggers prosurvival signaling and contributes to cell survival, invasive motility, and chemoresistance in many kinds of cancers. In addition, recent reports suggested that MerTK could be a primary target for abnormal platelet aggregation. Cons...

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Pubblicato in:Int J Mol Sci
Autori principali: Park, Tae Hyun, Bae, Seung-Hyun, Bong, Seoung Min, Ryu, Seong Eon, Jang, Hyonchol, Lee, Byung Il
Natura: Artigo
Lingua:Inglês
Pubblicazione: MDPI 2020
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7660649/
https://ncbi.nlm.nih.gov/pubmed/33114206
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/ijms21217878
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