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Crystal Structure of the Kinase Domain of MerTK in Complex with AZD7762 Provides Clues for Structure-Based Drug Development

Aberrant tyrosine-protein kinase Mer (MerTK) expression triggers prosurvival signaling and contributes to cell survival, invasive motility, and chemoresistance in many kinds of cancers. In addition, recent reports suggested that MerTK could be a primary target for abnormal platelet aggregation. Cons...

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Detalles Bibliográficos
Publicado en:Int J Mol Sci
Main Authors: Park, Tae Hyun, Bae, Seung-Hyun, Bong, Seoung Min, Ryu, Seong Eon, Jang, Hyonchol, Lee, Byung Il
Formato: Artigo
Idioma:Inglês
Publicado: MDPI 2020
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC7660649/
https://ncbi.nlm.nih.gov/pubmed/33114206
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/ijms21217878
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