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Romidepsin (FK228) and its analogs directly inhibit phosphatidylinositol 3‐kinase activity and potently induce apoptosis as histone deacetylase/phosphatidylinositol 3‐kinase dual inhibitors

Activation of phosphatidylinositol 3‐kinase (PI3K) signaling is involved in carcinogenesis and cancer progression. The PI3K inhibitors are considered candidate drugs for cancer treatment. Here, we describe a drug screening system for novel PI3K inhibitors using Saccharomyces cerevisiae strains with...

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Bibliografiske detaljer
Udgivet i:Cancer Sci
Main Authors: Saijo, Ken, Katoh, Tadashi, Shimodaira, Hideki, Oda, Akifumi, Takahashi, Ohgi, Ishioka, Chikashi
Format: Artigo
Sprog:Inglês
Udgivet: John Wiley and Sons Inc. 2012
Fag:
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC7659383/
https://ncbi.nlm.nih.gov/pubmed/22924958
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1111/cas.12002
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