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Pyrazolyl-pyrimidones inhibit the function of human solute carrier protein SLC11A2 (hDMT1) by metal chelation

Solute carrier proteins (SLCs) control fluxes of ions and molecules across biological membranes and represent an emerging class of drug targets. SLC11A2 (hDMT1) mediates intestinal iron uptake and its inhibition might be used to treat iron overload diseases such as hereditary hemochromatosis. Here w...

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Dettagli Bibliografici
Pubblicato in:RSC Med Chem
Autori principali: Poirier, Marion, Pujol-Giménez, Jonai, Manatschal, Cristina, Bühlmann, Sven, Embaby, Ahmed, Javor, Sacha, Hediger, Matthias A., Reymond, Jean-Louis
Natura: Artigo
Lingua:Inglês
Pubblicazione: Royal Society of Chemistry 2020
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7649969/
https://ncbi.nlm.nih.gov/pubmed/33479694
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/d0md00085j
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