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Optimal His-Tag Design for Efficient [(99m)Tc(CO)(3)](+) and [(188)Re(CO)(3)](+) Labeling of Proteins for Molecular Imaging and Radionuclide Therapy by Analysis of Peptide Arrays

Hexahistidine tags (His-tags), incorporated into recombinant proteins to facilitate purification using metal-affinity chromatography, are useful binding sites for radiolabeling with [(99m)Tc(CO)(3)](+) and [(188)Re(CO)(3)](+) for molecular imaging and radionuclide therapy. Labeling efficiencies vary...

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Publicat a:Bioconjug Chem
Autors principals: Williams, Jennifer D., Kampmeier, Florian, Badar, Adam, Howland, Kevin, Cooper, Margaret S., Mullen, Gregory E. D., Blower, Philip J.
Format: Artigo
Idioma:Inglês
Publicat: 2021
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC7611356/
https://ncbi.nlm.nih.gov/pubmed/33241692
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.bioconjchem.0c00561
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