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Cyclic boronates as versatile scaffolds for KPC-2 β-lactamase inhibition
Klebsiella pneumoniae carbapenemase-2 (KPC-2) is a serine-β-lactamase (SBL) capable of hydrolysing almost all β-lactam antibiotics. We compare KPC-2 inhibition by vaborbactam, a clinically-approved monocyclic boronate, and VNRX-5133 (taniborbactam), a bicyclic boronate in late-stage clinical develop...
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| Publicat a: | RSC Med Chem |
|---|---|
| Autors principals: | , , , , , , |
| Format: | Artigo |
| Idioma: | Inglês |
| Publicat: |
Royal Society of Chemistry
2020
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| Matèries: | |
| Accés en línia: | https://ncbi.nlm.nih.gov/pmc/articles/PMC7536818/ https://ncbi.nlm.nih.gov/pubmed/33479650 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/c9md00557a |
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