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PKIS deep dive yields a chemical starting point for dark kinases and a cell active BRSK2 inhibitor

The Published Kinase Inhibitor Set (PKIS) is a publicly-available chemogenomic library distributed to more than 300 laboratories by GlaxoSmithKline (GSK) between 2011 and 2015 and by SGC-UNC from 2015 to 2017. Screening this library of well-annotated, published kinase inhibitors has yielded a pletho...

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Bibliographic Details
Published in:Sci Rep
Main Authors: Tamir, Tigist Y., Drewry, David H., Wells, Carrow, Major, M. Ben, Axtman, Alison D.
Format: Artigo
Language:Inglês
Published: Nature Publishing Group UK 2020
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Online Access:https://ncbi.nlm.nih.gov/pmc/articles/PMC7522982/
https://ncbi.nlm.nih.gov/pubmed/32985588
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/s41598-020-72869-9
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