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AT101 [(-)-Gossypol] Selectively Inhibits MCL1 and Sensitizes Carcinoma to BH3 Mimetics by Inducing and Stabilizing NOXA

Anti-apoptotic BCL2 proteins are important targets for cancer therapy as cancers depend on their activity for survival. Direct inhibitors of MCL1 have entered clinical trials, although their efficacy may be limited by toxicity. An alternative approach may be to induce the pro-apoptotic protein NOXA...

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Dettagli Bibliografici
Pubblicato in:Cancers (Basel)
Autori principali: Mallick, David J., Eastman, Alan
Natura: Artigo
Lingua:Inglês
Pubblicazione: MDPI 2020
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7464284/
https://ncbi.nlm.nih.gov/pubmed/32824203
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/cancers12082298
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