Loading...

Tubulysin Synthesis Featuring Stereoselective Catalysis and Highly Convergent Multicomponent Assembly

[Image: see text] A concise and modular total synthesis of the highly potent N(14)-desacetoxytubulysin H (1) has been accomplished in 18 steps in an overall yield of up to 30%. Our work highlights the complexity–augmenting and route-shortening power of diastereoselective multicomponent reaction (MCR...

Fuld beskrivelse

Na minha lista:
Bibliografiske detaljer
Udgivet i:Org Lett
Main Authors: Vishwanatha, Thimmalapura M., Giepmans, Ben, Goda, Sayed K., Dömling, Alexander
Format: Artigo
Sprog:Inglês
Udgivet: American Chemical Society 2020
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC7372561/
https://ncbi.nlm.nih.gov/pubmed/32584589
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.orglett.0c01718
Tags: Tilføj Tag
Ingen Tags, Vær først til at tagge denne postø!