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Phase I study of TAS-115, a novel oral multi-kinase inhibitor, in patients with advanced solid tumors

TAS-115 is a novel MET, VEGFR, FMS and PDGFR inhibitor, developed to improve the continuity of drug administration with a relatively short half-life. We assessed its tolerability, safety, pharmacokinetics, efficacy, and pharmacodynamics in patients with solid tumors. This open-label, dose-escalation...

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Dettagli Bibliografici
Pubblicato in:Invest New Drugs
Autori principali: Doi, Toshihiko, Matsubara, Nobuaki, Kawai, Akira, Naka, Norifumi, Takahashi, Shunji, Uemura, Hiroji, Yamamoto, Noboru
Natura: Artigo
Lingua:Inglês
Pubblicazione: Springer US 2019
Soggetti:
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7340670/
https://ncbi.nlm.nih.gov/pubmed/31820255
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s10637-019-00859-4
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