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Abemaciclib induces atypical cell death in cancer cells characterized by formation of cytoplasmic vacuoles derived from lysosomes

In the cell cycle, the G(1)/S transition is controlled by the cyclin‐dependent kinase (CDK) 4/6‐cyclin D complex. Constitutive activation of CDK4/6 dysregulates G(1)/S transition, leading to oncogenic transformation. We found that 3 CDK4/6 inhibitors, abemaciclib, ribociclib, and palbociclib, exerte...

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Dettagli Bibliografici
Pubblicato in:Cancer Sci
Autori principali: Hino, Hirotsugu, Iriyama, Noriyoshi, Kokuba, Hiroko, Kazama, Hiromi, Moriya, Shota, Takano, Naoharu, Hiramoto, Masaki, Aizawa, Shin, Miyazawa, Keisuke
Natura: Artigo
Lingua:Inglês
Pubblicazione: John Wiley and Sons Inc. 2020
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7293084/
https://ncbi.nlm.nih.gov/pubmed/32304130
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1111/cas.14419
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