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Biased GPCR signaling: possible mechanisms and inherent limitations.

G protein-coupled receptors (GPCRs) are targeted by about a third of clinically used drugs. Many GPCRs couple to more than one type of heterotrimeric G proteins, become phosphorylated by any of several different GRKs, and then bind one or more types of arrestin. Thus, classical therapeutically activ...

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Bibliographische Detailangaben
Veröffentlicht in:Pharmacol Ther
Hauptverfasser: Gurevich, Vsevolod V., Gurevich, Eugenia V.
Format: Artigo
Sprache:Inglês
Veröffentlicht: 2020
Schlagworte:
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC7275904/
https://ncbi.nlm.nih.gov/pubmed/32201315
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.pharmthera.2020.107540
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