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Tamoxifen Directly Interacts with the Dopamine Transporter

The selective estrogen receptor modulator tamoxifen increases extracellular dopamine in vivo and acts as a neuroprotectant in models of dopamine neurotoxicity. We investigated the effect of tamoxifen on dopamine transporter (DAT)–mediated dopamine uptake, dopamine efflux, and [(3)H]WIN 35,428 [(–)-2...

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Detalles Bibliográficos
Publicado en:J Pharmacol Exp Ther
Autores principales: Mikelman, Sarah R., Guptaroy, Bipasha, Schmitt, Kyle C., Jones, Kymry T., Zhen, Juan, Reith, Maarten E. A., Gnegy, Margaret E.
Formato: Artigo
Lenguaje:Inglês
Publicado: The American Society for Pharmacology and Experimental Therapeutics 2018
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC7250473/
https://ncbi.nlm.nih.gov/pubmed/30108161
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/jpet.118.248179
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