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Design of gallinamide A analogs as potent inhibitors of the cysteine proteases human cathepsin L and Trypanosoma cruzi cruzain

Gallinamide A, originally isolated with modest antimalarial activity, was subsequently re-isolated and characterized as a potent, selective, and irreversible inhibitor of the human cysteine protease cathepsin L. Molecular docking identified potential modifications to improve binding, which were synt...

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Dettagli Bibliografici
Pubblicato in:J Med Chem
Autori principali: Boudreau, Paul D., Miller, Bailey W., McCall, Laura-Isobel, Almaliti, Jehad, Reher, Raphael, Hirata, Ken, Le, Thu, Siqueira-Neto, Jair L., Hook, Vivian, Gerwick, William H.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2019
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7240701/
https://ncbi.nlm.nih.gov/pubmed/31539239
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jmedchem.9b00294
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