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Pharmacology of tyrosine kinase inhibitors in chronic myeloid leukemia; a clinician’s perspective

OBJECTIVE: In this review, we have summarized the pharmacokinetics, pharmacodynamics and adverse effects of imatinib, dasatinib, nilotinib, bosutinib, ponatinib and radotinib with focus on pharmacogenomic studies with clinical end points. We have discussed the key phase 3 trials of tyrosine kinase i...

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Dettagli Bibliografici
Pubblicato in:Daru
Autori principali: Pushpam, Deepam, Bakhshi, Sameer
Natura: Artigo
Lingua:Inglês
Pubblicazione: Springer International Publishing 2020
Soggetti:
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7214547/
https://ncbi.nlm.nih.gov/pubmed/31900888
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s40199-019-00321-z
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