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Pharmacology of tyrosine kinase inhibitors in chronic myeloid leukemia; a clinician’s perspective

OBJECTIVE: In this review, we have summarized the pharmacokinetics, pharmacodynamics and adverse effects of imatinib, dasatinib, nilotinib, bosutinib, ponatinib and radotinib with focus on pharmacogenomic studies with clinical end points. We have discussed the key phase 3 trials of tyrosine kinase i...

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Bibliografski detalji
Izdano u:Daru
Glavni autori: Pushpam, Deepam, Bakhshi, Sameer
Format: Artigo
Jezik:Inglês
Izdano: Springer International Publishing 2020
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC7214547/
https://ncbi.nlm.nih.gov/pubmed/31900888
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s40199-019-00321-z
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