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Pharmacology of tyrosine kinase inhibitors in chronic myeloid leukemia; a clinician’s perspective

OBJECTIVE: In this review, we have summarized the pharmacokinetics, pharmacodynamics and adverse effects of imatinib, dasatinib, nilotinib, bosutinib, ponatinib and radotinib with focus on pharmacogenomic studies with clinical end points. We have discussed the key phase 3 trials of tyrosine kinase i...

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Detalhes bibliográficos
Publicado no:Daru
Main Authors: Pushpam, Deepam, Bakhshi, Sameer
Formato: Artigo
Idioma:Inglês
Publicado em: Springer International Publishing 2020
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC7214547/
https://ncbi.nlm.nih.gov/pubmed/31900888
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s40199-019-00321-z
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