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Receptor/gene/protein-mediated signaling connects methylprednisolone exposure to metabolic and immune-related pharmacodynamic actions in liver

A multiscale pharmacodynamic model was developed to characterize the receptor-mediated, transcriptomic, and proteomic determinants of corticosteroid (CS) effects on clinically relevant hepatic processes following a single dose of methylprednisolone (MPL) given to adrenalectomized (ADX) rats. The enh...

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Vydáno v:J Pharmacokinet Pharmacodyn
Hlavní autoři: Ayyar, Vivaswath S., Sukumaran, Siddharth, DuBois, Debra C., Almon, Richard R., Qu, Jun, Jusko, William J.
Médium: Artigo
Jazyk:Inglês
Vydáno: 2018
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC7167594/
https://ncbi.nlm.nih.gov/pubmed/29704219
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s10928-018-9585-x
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