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Perspective: Implications of Ligand–Receptor Binding Kinetics for Therapeutic Targeting of G Protein-Coupled Receptors

[Image: see text] The concept of ligand–receptor binding kinetics has been broadly applied in drug development pipelines focusing on G protein-coupled receptors (GPCRs). The ligand residence time (RT) for a receptor describes how long a ligand–receptor complex exists, and is defined as the reciproca...

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Veröffentlicht in:ACS Pharmacol Transl Sci
Hauptverfasser: van der Velden, Wijnand J. C., Heitman, Laura H., Rosenkilde, Mette M.
Format: Artigo
Sprache:Inglês
Veröffentlicht: American Chemical Society 2020
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC7155193/
https://ncbi.nlm.nih.gov/pubmed/32296761
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acsptsci.0c00012
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