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Discovering novel chemical inhibitors of human cyclophilin A: Virtual screening, synthesis, and bioassay

Cyclophilin A (CypA) is a member of cyclophilins, a family of the highly homologous peptidyl prolyl cis–trans isomerases (PPIases), which can bind to cyclosporin A (CsA). CypA plays critical roles in various biological processes, including protein folding, assembly, transportation, regulation of neu...

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Détails bibliographiques
Publié dans:Bioorg Med Chem
Auteurs principaux: Li, Jian, Chen, Jing, Gui, Chunshan, Zhang, Li, Qin, Yu, Xu, Qiang, Zhang, Jian, Liu, Hong, Shen, Xu, Jiang, Hualiang
Format: Artigo
Langue:Inglês
Publié: Elsevier Ltd. 2006
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC7119052/
https://ncbi.nlm.nih.gov/pubmed/16307882
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmc.2005.11.006
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