Caricamento...

Synthesis, biological evaluation and molecular modeling of novel azaspiro dihydrotriazines as influenza virus inhibitors targeting the host factor dihydrofolate reductase (DHFR)

Recently we identified cycloguanil-like dihydrotriazine derivatives, which provided host-factor directed antiviral activity against influenza viruses and respiratory syncytial virus (RSV), by targeting the human dihydrofolate reductase (hDHFR) enzyme. In this context we deemed interesting to further...

Descrizione completa

Salvato in:
Dettagli Bibliografici
Pubblicato in:Eur J Med Chem
Autori principali: Francesconi, Valeria, Giovannini, Luca, Santucci, Matteo, Cichero, Elena, Costi, Maria Paola, Naesens, Lieve, Giordanetto, Fabrizio, Tonelli, Michele
Natura: Artigo
Lingua:Inglês
Pubblicazione: Elsevier Masson SAS. 2018
Soggetti:
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7115377/
https://ncbi.nlm.nih.gov/pubmed/29886325
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.ejmech.2018.05.059
Tags: Aggiungi Tag
Nessun Tag, puoi essere il primo ad aggiungerne! !