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An efficient and tunable route to AG7088, a rhinovirus protease inhibitor

Aldol reaction of N,N-dibenzyl valinal with propiolic acid ethyl ester derived lithium reagent provides anti-aminoalcohol 8 and syn-aminoalcohol 9, which are converted into the lactone 6 via two different routes. Alkylation of 6 followed by lactone ring opening afford the acid 2a, which is coupled w...

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Dades bibliogràfiques
Publicat a:Tetrahedron Lett
Autors principals: Ma, Dawei, Xie, Weiqing, Zou, Bin, Lei, Qiong, Pei, Duanqing
Format: Artigo
Idioma:Inglês
Publicat: Elsevier Ltd. 2004
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC7111835/
https://ncbi.nlm.nih.gov/pubmed/32287436
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.tetlet.2004.08.179
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