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BIM-46174 fragments as potential ligands of G proteins

The 5,6,7,8-tetrahydroimidazo[1,2-a]pyrazine derivative BIM-46174 has received attention as Gα(q) inhibitor. We conducted structural reductions to monocyclic and bicyclic substructures to explore the chemical space of BIM fragments and to gain insights into the pharmacophore of BIM-type Gα(q) inhibi...

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Vydáno v:Medchemcomm
Hlavní autoři: Küppers, Jim, Benkel, Tobias, Annala, Suvi, Schnakenburg, Gregor, Kostenis, Evi, Gütschow, Michael
Médium: Artigo
Jazyk:Inglês
Vydáno: Royal Society of Chemistry 2019
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC7053702/
https://ncbi.nlm.nih.gov/pubmed/32180917
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/c9md00269c
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