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In silico Strategies to Support Fragment-to-Lead Optimization in Drug Discovery
Fragment-based drug (or lead) discovery (FBDD or FBLD) has developed in the last two decades to become a successful key technology in the pharmaceutical industry for early stage drug discovery and development. The FBDD strategy consists of screening low molecular weight compounds against macromolecu...
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| Publicat a: | Front Chem |
|---|---|
| Autors principals: | , , , , , , , |
| Format: | Artigo |
| Idioma: | Inglês |
| Publicat: |
Frontiers Media S.A.
2020
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| Matèries: | |
| Accés en línia: | https://ncbi.nlm.nih.gov/pmc/articles/PMC7040036/ https://ncbi.nlm.nih.gov/pubmed/32133344 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3389/fchem.2020.00093 |
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